Publications
Warren, GL; Do, TD; Kelley, BP; Nicholls, A; Warren, SD; “ESSENTIAL CONSIDERATIONS FOR USING PROTEIN-LIGAND STRUCTURES IN DRUG DISCOVERY”. Drug Discovery Today, (In Press)a,b
Warren, GL; Warren, SD; “SCORING DRUG-RECEPTOR INTERACTIONS”. Chapter 16 in Drug Design Strategies: Quantitative Approaches, Ed. by D. J. Livingstone and A. Davis, Royal Society of Chemistry, Cambridge, 2011, p. 440-457.b DOI:10.1039/9781849733410-00440
Warren, SD; “GUIDE TO FLUORINE NMR FOR ORGANIC CHEMISTS. BY WILLIAM R. DOLBIER, JR.” J. Med. Chem. 52, 6503, 2009.b
Grecian, SA; Hadida, S; Warren, SD; “DIRECT SYNTHESIS OF TRIMETHYL(2-PHENOXYETHYL)SILANES FROM AROMATIC FLUORIDES”. Tett. Lett. 46, 4683-4685, 2005.a
Trejo, A; Arzeno, H; Browner, M; Chanda, S; Cheng, S; Comer, DD; Dalrymple, SA; Dunten, P; Lafargue, J; Lovejoy, B; Freire-Moar, J; Lim, J; Mcintosh, J; Miller, J; Papp, E; Reuter, D; Roberts, R; Sanpablo, F; Saunders, J; Song, K; Villasenor, A; Warren, SD; Welch, M; Weller, P; Whiteley, PE; Zeng, L; and Goldstein, D; “DESIGN AND SYNTHESIS OF 4-AZAINDOLES AS INHIBITORS OF p38 MAP KINASE”. J. Med. Chem. 46, 4702-4713, 2003. a
Nair, SA; Kim, MH; Warren, SD; Choi, S; Songyang, Z; Cantley, LC; and Hangauer, DG; “IDENTIFICATION OF EFFICIENT PENTAPEPTIDE SUBSTRATES FOR THE TYROSINE KINASE pp60c-src”. J. Med. Chem. 38, 4276-4283, 1995. a
Warren, SD; “DESIGN, SYNTHESIS, ENZYME BINDING EVALUATION, AND ANALYSIS OF PREFERRED ENZYME-COMPLEXES FOR PEPTIDE-BASED cyclicAMP-DEPENDENT PROTEIN KINASE INHIBITORS”. Ph.D. Dissertation, State University of New York at Buffalo, 1995.c
Friedberg, JS; Tompkins, RG; Rakestraw, SL; Warren, SW; Fischman, AJ; and Yarmush, ML; "ANTIBODY-TARGETED PHOTOLYSIS: BACTERIOCIDAL EFFECTS OF Sn(IV) CHLORIN e6-DEXTRAN-MONOCLONAL ANTIBODY CONJUGATES". Ann. NY. Acad. Sci. 618, 383-393, 1991. a
Ali, SA; Warren, SD; Richter, KY; Badger, CC; Eary, JF; Press, OW; Krohn, KA; Bernstein, ID; and Nelp, WB; "IMPROVING THE TUMOR RETENTION OF RADIOIODINATED ANTIBODY: ARYL CARBOHYDRATE ADDUCTS". Cancer Res. 50, 783s-788s, 1990. a
Warren, SD; Ali, SA; Richter, KY; and Krohn, KA; "SYNTHESIS AND RADIOIODINATION OF TEN ARYL-CARBOHYDRATE COMPOUNDS FOR LABELING MONOCLONAL ANTIBODIES". J. Label. Comp. Radiopharm. 28, 497-509, 1990. a
Ali, SA; Eary, JF; Warren, SD; Badger, CC; and Krohn, KA; "SYNTHESIS AND RADIOIODINATION OF TYRAMINE CELLOBIOSE FOR LABELING MONOCLONAL ANTIBODIES". Nucl. Med. Biol. 15, 557-561, 1988 Int. J. Radiat. Appl. Instrum. Part B. a
"a" -Peer Reviewed; "b" -Editor Solicited/Invited, Editor Reviewed; "c" -Department Reviewed
ABSTRACTS & PRESENTATIONS
Warren, SD; Knapp, NR; Carlson, MA; Shelby, CA; Maul-Newby, HM; Watson, JM; Cronk, JD; “NEW ALLOSTERIC SITE INHIBITORS OF EUBACTERIAL β-CARBONIC ANHYDRASES”. NorthWest Crystallography Workshop, Bozeman, MT, July 20-22, 2012
Engerman, EM; Miller, CM; Warren, SD; “REACTIVITY OF THE EXOCYCLIC NITROGENS’ OF 2,4,6-TRIAMINOPYRIMIDINE”. Gonzaga’s Fall Family Weekend, Spokane, WA, October 21-23, 2011
Schwenne, KJ; Warren, SD; “ PROGRESS TOWARD THE SYNTHESIS OF 3-(4-BROMO-1h-IMIDAZOL-5-YL)PROPANEHYDROXAMIC ACID”. 66th Northwest Regional Meeting of the ACS, Portland, OR, June 26-29, 2011
Miller,CM; Carlson, MA; Knapp, NR; Sachet, ML; Langfield, A; Holden, J; Cronk, JD; Watson, J; Warren, SD; “LEAD GENERATION FOR POTENTIAL ALLOSTERIC INHIBITORS OF β–CARBONIC ANHYDRASE AND SYNTHESIS OF SUBSTITUTED PYRIMIDINE INHIBITORS”. Oral presentation at the 19th Regional Conference on Undergraduate Research Murdock College Science Research Program, Linfield College, McMinnville, OR, November 12 & 13, 2010
Miller,CM; Carlson, MA; Sachet, ML; Cronk, JD; Watson, J; Warren, SD; “SYNTHESIS OF SUBSTITUTED PYRIMIDINES AS INHIBITORS OF β–CARBONIC ANHYDRASE IN ESCHERICHIA COLI”. Presented at the 19th Regional Conference on Undergraduate Research Murdock College Science Research Program, Linfield College, McMinnville, OR, November 12 & 13, 2010
Carlson, MA; Knapp, NR; Sachet, ML; Langfield, A; Holden, J; Cronk, JD; Watson, J; Warren, SD; “LEAD GENERATION FOR POTENTIAL ALLOSTERIC INHIBITORS OF β–CARBONIC ANHYDRASE”. Presented at the 19th Regional Conference on Undergraduate Research Murdock College Science Research Program, Linfield College, McMinnville, OR, November 12 & 13, 2010
Warren, GL; Do, T; Warren, SD; “Iridium: Prepping PDB data for use in computation chemistry software development”. Presented at the 240th ACS National Meeting, Boston, MA, United States, August 22-26, 2010
Do, TD; Levingston, AL; Warren, SD; “Sequential one-pot syntheses of thiazoles and imidazo[2,1-b]thiazoles from amines, isothiocyanates and phenacyl bromides”. Presented at the Joint 65th Northwest and 22nd Rocky Mountain Regional Meeting of the American Chemical Society, Pullman, WA, United States, June 20-23, 2010
Knapp, NR; Holden, J; Carlson, MA; Warren, SD; Sachet, ML; Miller, CM; Watson, J; Langfield, A; Cronk, JD. “LEAD GENERATION FOR POTENTIAL ALLOSTERIC INHIBITORS OF β-CARBONIC ANHYDRASE”. Presented at the Joint 65th Northwest and 22nd Rocky Mountain Regional Meeting of the American Chemical Society, Pullman, WA, United States, June 20-23, 2010
Knapp, NR; Sachet, ML; Langfield, A; Holden, J; Cronk, JD; Watson, J; Warren, SD; “LEAD GENERATION FOR POTENTIAL ALLOSTERIC INHIBITORS OF β-CARBONIC ANHYDRASE”. Presented at the 18th Regional Conference on Undergraduate Research Murdock College Science Research Program, Gonzaga University, Spokane, WA, October 30-31, 2009.
Do, TD; Warren, GL; Warren, SD; “IRIDIUM: A CURATED DATABASE OF LIGAND-RECEPTOR COMPLEXES AND BINDING DATA”. Presented at the 18th Regional Conference on Undergraduate Research Murdock College Science Research Program, Gonzaga University, Spokane, WA, October 30-31, 2009.
Goossen, EA; Knapp, NR; Yee, DTt; Rhoads, T; Vadnais, K; Wisecup, A; Warren, SD; “SYNTHESIS OF 2,3-DIBENZYL-1,1-DIFLUOROGLYCEROL”. Presented at the 18th Regional Conference on Undergraduate Research Murdock College Science Research Program, Gonzaga University, Spokane, WA, October 30-31, 2009.
Oplinger, SL; Vadnais, KR; Warren, SD; “SPECTROPHOTOMETRIC ASSAYS OF LACTATE DEHYDROGENASE ACTIVITY IN THE PRESENCE OF LACTATE MIMETICS”. Presented at the 18th Regional Conference on Undergraduate Research Murdock College Science Research Program, Gonzaga University, Spokane, WA, October 30-31, 2009.
Knapp, NR; Sachet, ML; Langfield, A; Holden, J; Cronk, JD; Watson, J; Warren, SD; “LEAD GENERATION FOR POTENTIAL ALLOSTERIC INHIBITORS OF β-CARBONIC ANHYDRASE”. Presented at the 8th International Conference on Carbonic Anhydrases, Florence, Italy, September 16-19, 2009
Watson, J; Warren, SD; Knapp, NR; Langfield, A; Sachet, ML; Cronk, JD; “COMPUTATIONAL AND KINETIC CHARACTERIZATION OF THE ALLOSTERIC SITE IN E. COLI CARBONIC ANHYDRASE”. Presented at the 8th International Conference on Carbonic Anhydrases, Florence, Italy, September 16-19, 2009
Warren, GL; Do, TD; Warren, SD; “OF THINGS THAT ARE RARE: IRIDIUM, DINOSAUR COPROLITE, AND HIGH QUALITY PROTEIN-LIGAND STRUCTURE DATABASES”. Presented at the 238th ACS National Meeting, Washington, DC, August 16-20, 2009
Goossen, EA; Yee, DTt; Rhoads, TW; Vadnais, KR; Wisecup, A; Warren, SD; “SYNTHESIS OF 3,3-DIFLUORO-3-DEOXYGLYCEROL”. Presented at the 238th ACS National Meeting, Washington, DC, August 16-20, 2009
Goossen, EA; Yee, DTt; Rhoads, T; Vadnais, K; Wisecup, A; Warren, SD; “SYNTHESIS OF 2,3-DIBENZYL-1,1-DIFLUOROGLYCEROL”. Presented at the 64th Northwest Regional Meeting of the American Chemical Society, NW-140, Tacoma, WA, June 28-July 1, 2009.
Do, TD; Warren, GL; Warren, SD; “IRIDIUM: A CURATED DATABASE OF LIGAND-RECEPTOR COMPLEXES AND BINDING DATA”. Presented at the 64th Northwest Regional Meeting of the American Chemical Society, NW-140, Tacoma, WA, June 28-July 1, 2009.
Knapp, N; Cronk, JD; Warren, SD; “VIRTUAL SCREENING USED TO FIND POTENTIAL ALLOSTERIC INHIBITORS OF BETA-CARBONIC ANHYDRASE”. Presented at the 64th Northwest Regional Meeting of the American Chemical Society, NW-140, Tacoma, WA, June 28-July 1, 2009.
Do, T; Warren, GL; Warren, SD; “IRIDIUM: A CURATED DATABASE OF LIGAND-RECEPTOR COMPLEXES AND BINDING DATA”. Presented at CUP X, Santa Fe, New Mexico, March 8-11, 2009
Goossen, EA; Yee, DTt; Rhoads, T; Vadnais, K; Wisecup, A; Warren, SD; “SYNTHESIS OF 2,3-DIBENZYL-1,1-DIFLUOROGLYCEROL”. Presented at 17th Regional Conference on Undergraduate Research Murdock College Science Research Program, University of Puget Sound, Tacoma, WA, November 7-8, 2008
Knapp, N; Warren, SD; “VIRTUAL SCREENING USED TO FIND POTENTIAL ALLOSTERIC INHIBITORS OF BETA-CARBONIC ANHYDRASE”. Presented at 17th Regional Conference on Undergraduate Research Murdock College Science Research Program, University of Puget Sound, Tacoma, WA, November 7-8, 2008
Do, T; Warren, GL; Warren, SD; “A CURATED DATABASE OF LIGAND-RECEPTOR COMPLEXES AND THEIR BINDING DATA”. Presented at 17th Regional Conference on Undergraduate Research Murdock College Science Research Program, University of Puget Sound, Tacoma, WA, November 7-8, 2008
Goossen, E; Yee, DTt; Warren, SD;